Approved

Cosyntropin: Uses, Mechanism, and Reported Side Effects

Molecular formulaC136H210N40O31S
Molecular weight2933.4 g/mol
Registered trials96
PubChem CID16129617
Drug classAdrenocorticotropic Hormone [EPC]
Brand namesCosyntropin

If a doctor has ordered testing for possible adrenal insufficiency, cosyntropin may be part of that workup. It is a diagnostic agent, not a treatment, and its role is narrowly defined by its FDA label.

Key takeaways

  • Cosyntropin is classified as an adrenocorticotropic hormone used for diagnostic testing.
  • It is approved to help screen for adrenocortical insufficiency by measuring plasma cortisol response.
  • The approved brand name is Cosyntropin.
  • Over 90 registered trials have studied cosyntropin or involved it as a testing tool.
  • Reported adverse events span pregnancy-related exposure reports, low blood sugar, low blood pressure, and respiratory symptoms.

What Cosyntropin Is

Cosyntropin belongs to a drug class known as adrenocorticotropic hormones. It is a synthetic compound built to act like the natural hormone that signals the adrenal glands. Its identity is catalogued under PubChem CID 16129617.

What Cosyntropin Is Approved For

Cosyntropin is approved as a diagnostic agent to screen patients suspected of having adrenocortical insufficiency. It works by prompting a rapid adrenal cortex response, allowing clinicians to measure plasma cortisol over a short test window, often around 30 minutes, using just two blood draws. The label notes that a normal basal cortisol level does not rule out insufficiency, since some patients only show abnormal responses under stress. No boxed warning is present on the label. The approved brand is marketed as Cosyntropin.

What the Evidence Shows

Clinical trial registries list 96 studies connected to cosyntropin, though many use it as a diagnostic or research tool rather than as the primary intervention. A completed Phase 2 trial examined dexamethasone for preventing oral chronic graft-versus-host disease, incorporating cosyntropin-based adrenal assessment. A separate early-phase trial exploring longer-term adrenal suppression with low-dose hydrocortisone was withdrawn before completion.

Reported Side Effects

Adverse event reports submitted to FAERS reflect counts of reported reactions, not confirmed incidence or direct causation. The most frequently reported issues relate to pregnancy exposure, including foetal growth restriction (24 reports) and foetal exposure during pregnancy (23 reports). Metabolic and cardiovascular reactions also appear, including hypoglycaemia (20), hypotension (18), and hyperkalaemia (11). Respiratory and general reactions include dyspnoea and pneumonia (13 reports each), along with nausea (12 reports).

FAQ

What is cosyntropin used for?
Cosyntropin is an FDA-approved diagnostic agent used to screen patients suspected of having adrenocortical insufficiency. It measures how well the adrenal cortex responds by tracking plasma cortisol levels after administration. It is used for testing purposes only, not as a treatment.
How does cosyntropin work?
Cosyntropin acts on the adrenal cortex to trigger a rapid cortisol response, which clinicians can measure using blood samples taken shortly after administration. This response helps distinguish normal adrenal function from insufficiency. The label notes this test can often be completed within about 30 minutes.
Does a normal basal cortisol level rule out adrenal insufficiency?
No. The label specifically states that a normal basal cortisol level does not by itself rule out adrenal insufficiency. Some patients with proven insufficiency have normal baseline levels and only show abnormal responses when stressed, which is part of why the cosyntropin test is useful.
What side effects have been reported with cosyntropin?
Reported reactions include pregnancy-related events such as foetal growth restriction and foetal exposure during pregnancy, along with hypoglycaemia, hypotension, and hyperkalaemia. Dyspnoea, pneumonia, and nausea have also been reported. These are counts of submitted reports, not confirmed rates or proof that cosyntropin caused the reaction.
Does cosyntropin carry a boxed warning?
No, the current label for cosyntropin does not carry a boxed warning.
This page is an editorial information resource. It does not sell, prescribe, or recommend any medication. Content is editorial information, not medical advice. Talk to your doctor before any treatment decision.

Sources: FDA drug label (DailyMed) PubChem ClinicalTrials.gov FDA Adverse Event Reporting System (FAERS)

Updated 2026-09-19